ACS MEDI division news
ResMed: Residential School on Medicinal Chemistry and Biology in Drug Discovery
ResMed is a week-long graduate level course organized to provide an accelerated program for medicinal chemists, biologists and other industrial and academic scientists who wish to broaden their knowledge of drug discovery and development. The School’s aim is to concentrate on the fundamentals that are useful in drug discovery spanning initial target validation through development.
TOPICS INCLUDE
Principles of Med Chem
Drug-like Properties
Hit-to-Lead in Drug Discovery
Lead Optimization Cheminformatics
Molecular Modeling & Structure-Based Drug Design Kinases
Drug Metabolism
Designing Around Problematic Functionalities Bioisosteres
Covalent Inhibitors Pharmacokinetics & Protein Binding Enzymology, Receptors & Ion Channels Proximity-induced Drug Design Proteolysis-targeting Chimeras Phenotypic Screening Protein-protein interactions Antibody-drug Conjugates
Preclinical Toxicology
In Silico Tools
Impact of AI
Case Study Presentations